About 30 results found for searched term "Dopamine Receptor" (0.063 seconds)
| Cat.No. | Name | Target |
|---|---|---|
| M2349 | (R)-Nepicastat hydrochloride | HCV Protease |
| RS-25560-198 HCl | ||
| (R)-Nepicastat hydrochloride, the R-enantiomer of Nepicastat hydrochloride, is a potent and selective inhibitor with IC50 of 25.1 nM and 18.3 nM for bovine and human dopamine-β-hydroxylase, with negligible affinity for twelve other enzymes and thirteen neurotransmitter receptors. | ||
| M2372 | Alizapride hydrochloride | Dopamine Receptor |
| Alizapride hydrochloride is a dopamine receptor antagonist used for the theropy of nausea and vomiting. | ||
| M2494 | Cariprazine hydrochloride | Dopamine Receptor |
| RGH-188 HCl | ||
| Cariprazine hydrochloride is a dopamine D3-receptor-preferring partial agonist that exhibits high selectivity and affinity to dopamine D3 and D2(L/S) receptors with pKi 10.07 and 9.16/9.31, respectively. | ||
| M2655 | Droperidol | Dopamine Receptor |
| Dehydrobenzperidol | ||
| Droperidol is a potent antagonist of dopamine subtype 2 receptors in the limbic system. | ||
| M2886 | Nomifensine Maleate | Dopamine Receptor |
| (±)-Nomifensine maleat | ||
| Nomifensine is a dopamine reuptake inhibitor that increases the amount of synaptic dopamine available to receptors by blocking dopamine's re-uptake transporter. | ||
| M2936 | Phenothiazine | Dopamine Receptor |
| Phenothiazine is a dopamine-2 (D2) receptor antagonist therefore decreases the effect of dopamine in the brain. | ||
| M2987 | Ropinirole hydrochloride | Dopamine Receptor |
| SKF 101468 hydrochloride | ||
| Ropinirole a selective dopamine D2 receptors inhibitor with IC50 of 29 nM. | ||
| M3065 | Thioridazine hydrochloride | Dopamine Receptor |
| Thioridazine is a trifluoro-methyl phenothiazine derivative, which blocks postsynaptic mesolimbic dopaminergic D1 and D2 receptors in the brain. | ||
| M3087 | Trifluoperazine dihydrochloride | Dopamine Receptor |
| TFP; SKF5019 | ||
| Trifluoperazine is a dopamine D2 receptor inhibitor with IC50 of 1.1 nM. | ||
| M3088 | Triflupromazine hydrochloride | Dopamine Receptor |
| Triflupromazine hydrochloride is a member of a family of phenothiazine compounds that are dopamine D1/D2 receptor antagonists. | ||
| M3165 | Prochlorperazine dimaleate | Dopamine Receptor |
| Prochlorperazine dimaleate is a D2 dopamine receptor antagonist. | ||
| M3242 | Sumanirole Maleate | Dopamine Receptor |
| U 95666E | ||
| Sumanirole maleate is a highly selective dopamine D2 receptor agonist with binding affinity of 9 nM and EC50 of about 46 nM, exhibits >200-fold selectivity over the other dopamine receptor subtypes. | ||
| M3287 | PD128907 hydrochloride | Dopamine Receptor |
| PD 128907 hydrochloride is a potent and selective dopamine D3 receptor agonist, with EC50 of 0.64 nM, exhibits 53-fold selectivity over dopamine D2 receptor. | ||
| M3320 | Quetiapine Fumarate | 5-HT Receptor |
| Quetiapine hemifumarate | ||
| Quetiapine hemifumarate is a 5-HT receptors agonist with a pEC50 of 4.77 for human 5-HT1A receptor. Quetiapine hemifumarate is a dopamine receptor antagonist with a pIC50 of 6.33 for human D2 receptor. | ||
| M3414 | Olanzapine | 5-HT Receptor |
| LY170053 | ||
| Olanzapine is a high affinity for 5-HT2 serotonin and D2 dopamine receptor antagonist. | ||
| M3479 | Aripiprazole | 5-HT Receptor |
| OPC-14597 | ||
| Aripiprazole is a human 5-HT1A receptor partial agonist with a Ki of 4.2 nM. Aripiprazole (OPC-14597) is a potent and high-affinity dopamine D2 receptor partial agonist. | ||
| M3481 | WAY-100635 Maleate | 5-HT Receptor |
| WAY-100635 maleate is a potent, selective 5-HT1A receptor antagonist with an IC50 value of 0.91 nM, a Ki value of 0.39 nM, and a pIC50 of 8.87, which is more than 100-fold more selective than for use at the other 5-HT receptor subtypes and major neurotransmitter receptors. In addition, WAY-100635 maleate is a potent dopamine D4 receptor agonist. | ||
| M3592 | Chlorprothixene | Dopamine Receptor |
| Chlorprothixene has strong binding affinities to dopamine and histamine receptors, such as D1, D2, D3, D5, H1, 5-HT2, 5-HT6 and 5-HT7, with Ki of 18 nM, 2.96 nM, 4.56 nM, 9 nM, 3.75 nM, 9.4 nM, 3 nM and 5.6 nM, respectively. | ||
| M3670 | Metoclopramide hydrochloride | 5-HT Receptor |
| Metoclopramide hydrochloride is a selective dopamine D2 receptor antagonist, used for the treatment of nausea and vomiting. | ||
| M3675 | Rotigotine | Dopamine Receptor |
| N-0923 | ||
| Rotigotine is a potent dopamine receptor agonist with Ki values of 0.71 nM, 4-15 nM, and 83 nM for the dopamine D3 receptor and D2, D5, D4 receptors and dopamine D1 receptor. Rotigotine a partial agonist of the 5-HT1A receptor, and an antagonist of the α2B-adrenergic receptor. | ||
| M3785 | Flupenthixol dihydrochloride | Dopamine Receptor |
| Flupenthixol 2HCl | ||
| Flupenthixol dihydrochloride is a dopamine receptor antagonist which acts as a Neuroleptic agent as well as an antipsychotic. | ||
| M3818 | Rotigotine Hydrochloride | Dopamine Receptor |
| Rotigotine HCl;N-0923 Hydrochloride | ||
| Rotigotine Hydrochloride (N-0923 Hydrochloride) is a full agonist of dopamine receptor, a partial agonist of the 5-HT1A receptor, and an antagonist of the α2B-adrenergic receptor, with Ki of 0.71 nM, 4-15 nM, and 83 nM for the dopamine D3 receptor and D2, D5, D4 receptors, and dopamine D1 receptor. | ||
| M1565 | Quetiapine sulfoxide | 5-HT Receptor |
| Quetiapine sulfoxide; Quetiapine S-oxide | ||
| Quetiapine sulfoxide is a 5-HT receptor agonist with a pEC50 value of 4.77 for human 5-HT1A. Quetiapine hemifumarate is a dopamine receptor antagonist with a pIC50 value of 6.33 for human D2. | ||
| M1564 | Quetiapine Sulfone | 5-HT Receptor |
| Quetiapine Sulfone is a 5-HT receptor agonist with a pEC50 value of 4.77 for human 5-HT1A. Quetiapine hemifumarate is a dopamine receptor antagonist with a pIC50 value of 6.33 for human D2. | ||
| M1454 | Buspirone | 5-HT Receptor |
| Buspirone is an orally active 5-HT1A receptor agonist, and a dopamine D2 autoreceptorsant antagonist. | ||
| M4458 | Tetrahydroberberine | Dopamine Receptor |
| Canadine; THB | ||
| Tetrahydroberberine is an isoquinoline alkaloid isolated from corydalis tuber; has micromolar affinity for dopamine D(2) (pK(i) = 6.08) and 5-HT(1A) (pK(i) = 5.38) receptors but moderate to no affinity for other relevant serotonin receptors (5-HT(1B), 5-HT(1D), 5-HT(3), and 5-HT(4); pK(i) < 5.00). | ||
| M4887 | Pardoprunox Hydrochloride | 5-HT Receptor |
| SLV-308 | ||
| Pardoprunox hydrochloride (DU-126891, SME-308) is an effective agonist of partial dopamine action, corresponding to pEC50 value 8.0. It is also a partial agonist inducing [35S]GTPγS binding, corresponding to pEC50 9.2 and serotonin 5-HT1A receptor 6.3. | ||
| M5424 | Asenapine maleate | 5-HT Receptor |
| Org 5222 | ||
| Asenapine maleate is a high-affinity antagonist of various receptors including serotonin receptors (5-HT), norepinephrine (NA), dopamine receptors, and histamine receptors, and can be used in studies related to neurodivergent disorders as well as depressive manic depression. | ||
| M5456 | B-HT 920 dihydrochloride | Adrenergic Receptor |
| Talipexole dihydrochloride | ||
| B-HT 920(Talipexole 2Hcl) is a dopamine D2 receptor agonist, α2-adrenoceptor agonist and 5-HT3 receptor antagonist, which displays antiParkinsonian activity. | ||
| M5467 | Brexpiprazole | Dopamine Receptor |
| OPC-34712, OPC 34712, OPC34712 | ||
| Brexpiprazole is a novel D2 dopamine and serotonin 1A partial agonist, called serotonin-dopamine activity modulator (SDAM), and a potent antagonist of serotonin 2A receptors, noradrenergic alpha 1B and 2C receptors. | ||
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